SS-31

Also known as: Elamipretide, Bendavia, MTP-131

A mitochondria-targeted peptide for cellular energy and tissue protection.

Overview

SS-31 is a cell-permeable tetrapeptide that selectively concentrates in the inner mitochondrial membrane. It protects mitochondrial function and has shown promise in conditions involving mitochondrial dysfunction.

Mechanism of Action

Binds cardiolipin in the inner mitochondrial membrane, stabilizing cristae structure and optimizing electron transport chain function. Reduces ROS production and prevents cytochrome c release.

Pharmacokinetics

Rapid cellular uptake with mitochondrial targeting. Half-life approximately 4 hours.

Dosing Protocols

Note: These are research protocols from literature. This is not medical advice.

1

Standard

Dose

40 mg

Frequency

Once daily

Duration

4-8 weeks

Clinical trial dosing

2

Research

Dose

0.25-0.5 mg/kg

Frequency

Once daily

Duration

Variable

Preclinical extrapolation

Stacking Recommendations

Peptides that may be combined based on complementary mechanisms in research settings.

Rationale: Mitochondrial support

Synergy: Dual mitochondrial optimization

Rationale: Cellular health

Synergy: Comprehensive cellular protection

Research Areas

Heart FailureMitochondrial DiseasesKidney DiseaseAge-Related Conditions

Key Research Findings

  • 1Improved cardiac function in heart failure trials
  • 2Reduced kidney injury in ischemia models
  • 3Enhanced exercise capacity in mitochondrial myopathy
  • 4Protected neurons in neurodegenerative models

Side Effects & Contraindications

Reported Side Effects

  • Injection site reactions
  • Headache

Contraindications

  • Pregnancy

Safety Considerations

Generally well-tolerated in clinical trials. Injection site reactions most common.

Storage Requirements

Store at 2-8C

Scientific References

Quick Reference

Sequence
D-Arg-Dmt-Lys-Phe-NH2
Molecular Weight
639 g/mol
Half-Life
~4 hours
Bioavailability
High (SC)
Research Stage
clinical phase 3
Administration
Subcutaneous or intravenous