ARA-290

Also known as: Cibinetide

An erythropoietin-derived peptide for tissue protection without erythropoietic effects.

Overview

ARA-290 is an 11-amino acid peptide derived from the tissue-protective region of erythropoietin. It activates the innate repair receptor without stimulating red blood cell production.

Mechanism of Action

Activates the innate repair receptor (IRR), a heterodimer of EPO-R and CD131. Promotes tissue protection and repair through anti-inflammatory and anti-apoptotic pathways.

Pharmacokinetics

Short half-life requiring daily dosing. Good tissue distribution.

Dosing Protocols

Note: These are research protocols from literature. This is not medical advice.

1

Standard

Dose

4 mg

Frequency

Once daily

Duration

28 days

Clinical trial protocol

Stacking Recommendations

Peptides that may be combined based on complementary mechanisms in research settings.

Rationale: Neuroprotection

Synergy: Nerve healing support

Research Areas

NeuropathyChronic Kidney DiseaseDiabetic ComplicationsSarcoidosis

Key Research Findings

  • 1Improved small fiber neuropathy symptoms in clinical trials
  • 2Reduced neuropathic pain scores
  • 3Anti-inflammatory effects without erythropoiesis
  • 4Potential in diabetic complications

Side Effects & Contraindications

Reported Side Effects

  • Injection site reactions
  • Headache

Contraindications

  • Active malignancy

Safety Considerations

Well-tolerated in clinical trials. No erythropoietic effects observed.

Storage Requirements

Store at 2-8C

Scientific References

Quick Reference

Sequence
QEQLERALNSS
Molecular Weight
1258 g/mol
Half-Life
~1-2 hours
Bioavailability
High (SC)
Research Stage
clinical phase 2
Administration
Subcutaneous injection