PTD-DBM

Also known as: Protein Transduction Domain-DBM, Bone Formation Peptide

A cell-penetrating peptide for bone regeneration and fracture healing.

Overview

PTD-DBM is a synthetic peptide combining a protein transduction domain with a BMP-binding sequence. It enhances bone morphogenetic protein (BMP) signaling to promote bone formation and healing. It shows promise for fracture repair and bone regeneration.

Mechanism of Action

The PTD allows cell penetration while the DBM (demineralized bone matrix-binding) sequence enhances BMP-2 signaling. Promotes osteoblast differentiation and bone formation. May reduce the BMP dose needed for bone healing.

Pharmacokinetics

Local application to bone defects. Cell-penetrating peptide allows tissue uptake.

Dosing Protocols

Note: These are research protocols from literature. This is not medical advice.

1

Bone Healing Research

Dose

Variable

Frequency

Single or repeated local application

Duration

Until healing

Applied to fracture or defect site

Stacking Recommendations

Peptides that may be combined based on complementary mechanisms in research settings.

Rationale: Healing synergy

Synergy: Comprehensive tissue repair

Research Areas

Fracture HealingBone RegenerationOsteoporosisSpinal FusionDental ImplantsOrthopedics

Key Research Findings

  • 1Enhanced bone formation in animal models
  • 2Synergizes with BMPs for healing
  • 3Cell-penetrating delivery improves uptake
  • 4Potential to reduce BMP doses needed

Side Effects & Contraindications

Reported Side Effects

  • Local reactions
  • Limited systemic data

Contraindications

  • Active bone infection
  • Malignancy at site

Safety Considerations

Research compound. Local application. Limited systemic data. Used in orthopedic research settings.

Storage Requirements

Store at -20°C

Scientific References

Quick Reference

Sequence
PTD sequence + DBM binding domain
Molecular Weight
~2.5 kDa
Half-Life
Variable (local application)
Bioavailability
Local application
Research Stage
preclinical
Administration
Local injection or implant