Orexin B

Also known as: Hypocretin-2, OX-B, HCRT-2

A neuropeptide related to Orexin A, regulating sleep, arousal, and metabolism.

Overview

Orexin B (Hypocretin-2) is a 28-amino acid neuropeptide closely related to Orexin A. It is produced in the same hypothalamic neurons and plays similar roles in regulating sleep-wake cycles, arousal, and feeding behavior. It has slightly different receptor selectivity compared to Orexin A.

Mechanism of Action

Primarily activates OX2R (orexin receptor 2) with less activity at OX1R compared to Orexin A. Promotes wakefulness and arousal. Regulates feeding behavior and energy homeostasis.

Pharmacokinetics

Poor BBB penetration peripherally. Short half-life. Research typically uses intranasal or central delivery.

Dosing Protocols

Note: These are research protocols from literature. This is not medical advice.

1

Research

Dose

10-50 mcg

Frequency

As needed

Duration

Acute studies

Experimental only

Stacking Recommendations

Peptides that may be combined based on complementary mechanisms in research settings.

Rationale: Complete orexin system

Synergy: Both peptides work together naturally

Research Areas

NarcolepsySleep DisordersArousalAppetite RegulationMetabolismCognitive Function

Key Research Findings

  • 1Co-released with Orexin A from hypothalamic neurons
  • 2More selective for OX2R than Orexin A
  • 3Involved in sleep-wake regulation
  • 4Deficiency contributes to narcolepsy

Side Effects & Contraindications

Reported Side Effects

  • Anxiety
  • Increased alertness
  • Appetite changes
  • Cardiovascular effects

Contraindications

  • Anxiety disorders
  • Insomnia
  • Cardiovascular disease

Safety Considerations

Research compound. Limited safety data. May cause overstimulation, anxiety, or cardiovascular effects.

Storage Requirements

Store at -20°C

Scientific References

Quick Reference

Sequence
28 amino acid peptide
Molecular Weight
2937 g/mol
Half-Life
Minutes
Bioavailability
Poor peripheral, intranasal research
Research Stage
preclinical
Administration
Intranasal (research)