KPV

Also known as: Alpha-MSH Fragment, Lys-Pro-Val

An anti-inflammatory tripeptide derived from alpha-MSH with gut healing properties.

Overview

KPV is a tripeptide representing the C-terminal sequence of alpha-melanocyte stimulating hormone (a-MSH). It retains the anti-inflammatory properties of the parent molecule without melanogenic effects.

Mechanism of Action

Inhibits NF-kB and MAPK inflammatory pathways. Reduces pro-inflammatory cytokine production. Promotes intestinal epithelial healing and barrier function.

Pharmacokinetics

Small peptide with good tissue penetration. Can be administered orally for GI effects due to local action.

Dosing Protocols

Note: These are research protocols from literature. This is not medical advice.

1

Oral/Gut Health

Dose

200-500 mcg

Frequency

1-2 times daily

Duration

4-8 weeks

Oral capsule for IBD applications

2

Subcutaneous

Dose

200 mcg

Frequency

Once daily

Duration

4 weeks

Systemic anti-inflammatory

Stacking Recommendations

Peptides that may be combined based on complementary mechanisms in research settings.

Rationale: Gut healing synergy

Synergy: Dual mechanism GI protection and repair

Research Areas

Inflammatory Bowel DiseaseGut HealthSkin InflammationWound Healing

Key Research Findings

  • 1Reduced inflammation in colitis models
  • 2Improved intestinal barrier function
  • 3Decreased pro-inflammatory cytokines (TNF-a, IL-6, IL-1b)
  • 4Accelerated wound healing in skin models

Side Effects & Contraindications

Reported Side Effects

  • Generally well-tolerated

Contraindications

  • Pregnancy (insufficient data)

Safety Considerations

Generally well-tolerated. No significant adverse effects reported in studies.

Storage Requirements

Store at -20C or 2-8C

Scientific References

Quick Reference

Sequence
Lys-Pro-Val
Molecular Weight
342.43 g/mol
Half-Life
Short
Bioavailability
Good oral bioavailability for gut applications
Research Stage
preclinical
Administration
Oral, topical, or subcutaneous