GHRP-2

Featured

Also known as: Growth Hormone Releasing Peptide-2, Pralmorelin

A potent growth hormone secretagogue with strong GH-releasing effects.

Overview

GHRP-2 is one of the most potent synthetic GH secretagogues. It stimulates robust GH release through ghrelin receptor activation and is used diagnostically to assess GH reserve.

Mechanism of Action

Binds ghrelin receptors (GHS-R1a) on pituitary somatotrophs and hypothalamic neurons. Stimulates GH release and mildly increases cortisol and prolactin.

Pharmacokinetics

Rapid absorption with peak GH at 15-30 minutes. Effects last 2-3 hours. Half-life approximately 25-30 minutes.

Dosing Protocols

Note: These are research protocols from literature. This is not medical advice.

1

Standard

Dose

100-300 mcg

Frequency

2-3x daily

Duration

8-12 weeks

Best combined with GHRH

2

Diagnostic

Dose

1 mcg/kg IV

Frequency

Single dose

Duration

N/A

GH stimulation test

Stacking Recommendations

Peptides that may be combined based on complementary mechanisms in research settings.

Rationale: Maximum GH release

Synergy: Synergistic GHRH + GHRP

Rationale: Enhanced pulsatility

Synergy: Dual receptor activation

Research Areas

GH Deficiency TestingMuscle GrowthAnti-AgingAppetite Stimulation

Key Research Findings

  • 1Most potent GHRP for GH release
  • 2Approved in Japan for GH stimulation testing
  • 3Significant increases in IGF-1 with regular use
  • 4Appetite stimulation due to ghrelin pathway

Side Effects & Contraindications

Reported Side Effects

  • Increased appetite
  • Water retention
  • Elevated cortisol
  • Flushing

Contraindications

  • Prolactinoma
  • Active malignancy

Safety Considerations

Increases cortisol and prolactin (unlike ipamorelin). May stimulate appetite. Water retention possible.

Storage Requirements

Store lyophilized at -20C

Scientific References

Quick Reference

Sequence
D-Ala-D-2-Nal-Ala-Trp-D-Phe-Lys-NH2
Molecular Weight
817.97 g/mol
Half-Life
25-30 minutes
Bioavailability
High (SC)
Research Stage
approved
Administration
Subcutaneous or intravenous